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AKR1C3-IN-6

Catalog No. T61790Cas No. 2137881-54-8

AKR1C3-IN-6 (Compound 1) is a potent and specific AKR1C3 inhibitor, exhibiting IC50 values of 0.31 μM against AKR1C3 and 73.23 μM against AKR1C2. It demonstrates significant antitumor activity [1].

AKR1C3-IN-6

AKR1C3-IN-6

Catalog No. T61790Cas No. 2137881-54-8
AKR1C3-IN-6 (Compound 1) is a potent and specific AKR1C3 inhibitor, exhibiting IC50 values of 0.31 μM against AKR1C3 and 73.23 μM against AKR1C2. It demonstrates significant antitumor activity [1].
Pack SizePriceAvailabilityQuantity
25 mg$1,5208-10 weeks
50 mg$1,9808-10 weeks
100 mg$2,5008-10 weeks
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Product Introduction

Bioactivity
Description
AKR1C3-IN-6 (Compound 1) is a potent and specific AKR1C3 inhibitor, exhibiting IC50 values of 0.31 μM against AKR1C3 and 73.23 μM against AKR1C2. It demonstrates significant antitumor activity [1].
In vitro
Compound 1 (AKR1C3-IN-6) exhibits antiproliferative effects, demonstrating an IC50 value of 81.40 ± 2.29 μM against the 22rv1 prostate cancer cell line [1].
Chemical Properties
Molecular Weight392.33
FormulaC18H15F3N4O3
Cas No.2137881-54-8
Storage & Solubility Information
StorageShipping with blue ice.

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