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Apimostinel (NRX-1074; AGN-241660) is a partial agonist of the NMDA receptor.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $1,490 | 6-8 weeks | |
50 mg | $1,940 | 6-8 weeks | |
100 mg | $2,800 | 6-8 weeks |
Description | Apimostinel (NRX-1074; AGN-241660) is a partial agonist of the NMDA receptor. |
In vitro | Apimostinel (NRX-1074) modulates the NMDA receptor similarly to GLYX-13 but includes a synthetic amino acid modification that enhances its potency and oral bioavailability[1]. |
In vivo | In preclinical models, both compounds demonstrate high efficacy in treating various CNS disorders[1]. |
Alias | NRX-1074, AGN-241660 |
Molecular Weight | 503.59 |
Formula | C25H37N5O6 |
Cas No. | 1421866-48-9 |
Relative Density. | 1.330 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 155 mg/mL (307.79 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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