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Aurora inhibitor 1 is a potent inhibitor of Aurora A and Aurora B kinases with IC50 values of ≤ 4 nM and ≤ 13 nM, respectively.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $3,130 | 3-6 months | |
50 mg | $4,610 | 3-6 months | |
100 mg | $5,730 | 3-6 months |
Description | Aurora inhibitor 1 is a potent inhibitor of Aurora A and Aurora B kinases with IC50 values of ≤ 4 nM and ≤ 13 nM, respectively. |
Targets&IC50 | Aurora B:13 nM, Aurora A:4 nM |
In vitro | Aurora inhibitor 1 (Compound 16) demonstrates Kd values of 0.01 nM for both Aurora A and Aurora B kinases. |
In vivo | In vivo efficacy in a mouse xenograft tumor model when dosed orally, Aurora inhibitor 1 exhibits good drug exposure levels across species upon oral dosing and shows excellent. |
Molecular Weight | 459.57 |
Formula | C23H25N9S |
Cas No. | 2227019-45-4 |
Relative Density. | 1.41 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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