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BAY-252

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Catalog No. T78148Cas No. 2639638-67-6

BAY-252 is a potent inhibitor of branched-chain amino acid transaminases 1 (BCAT1) and BCAT2, demonstrating inhibitory concentration (IC50) values of 2 μM for both enzymes. Additionally, BAY-069 serves as a chemical probe and is applicable in cancer research [1].

BAY-252

BAY-252

😃Good
Catalog No. T78148Cas No. 2639638-67-6
BAY-252 is a potent inhibitor of branched-chain amino acid transaminases 1 (BCAT1) and BCAT2, demonstrating inhibitory concentration (IC50) values of 2 μM for both enzymes. Additionally, BAY-069 serves as a chemical probe and is applicable in cancer research [1].
Pack SizePriceAvailabilityQuantity
5 mgInquiry8-10 weeks
50 mgInquiry8-10 weeks
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Product Introduction

Bioactivity
Description
BAY-252 is a potent inhibitor of branched-chain amino acid transaminases 1 (BCAT1) and BCAT2, demonstrating inhibitory concentration (IC50) values of 2 μM for both enzymes. Additionally, BAY-069 serves as a chemical probe and is applicable in cancer research [1].
In vitro
BAY-252 inhibits the proliferation of MDA-MB-231 cells with an IC50 value of 2 μM [1].
Chemical Properties
Molecular Weight446.81
FormulaC22H14ClF3N2O3
Cas No.2639638-67-6
Storage & Solubility Information
StorageShipping with blue ice.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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