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BMS-986163

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Catalog No. T14686Cas No. 1801151-09-6

BMS-986163, a negative allosteric modulator of GluN2B, rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM) as a prodrug.

BMS-986163

BMS-986163

😃Good
Catalog No. T14686Cas No. 1801151-09-6
BMS-986163, a negative allosteric modulator of GluN2B, rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM) as a prodrug.
Pack SizePriceAvailabilityQuantity
25 mg$2,42010-14 weeks
50 mg$3,18010-14 weeks
100 mg$4,30010-14 weeks
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Product Introduction

Bioactivity
Description
BMS-986163, a negative allosteric modulator of GluN2B, rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM) as a prodrug.
Targets&IC50
GluN2B, BMS-986169:24 nM, GluN2B, BMS-986169:4 nM
Chemical Properties
Molecular Weight462.45
FormulaC23H28FN2O5P
Cas No.1801151-09-6
Relative Density.1.38 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Keywords

BMS986163BMS 986163BMS-986163
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