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Bosentan-d4

Catalog No. T73820Cas No. 1065472-77-6

Bosentan-d4, the deuterium-labeled variant of Bosentan, serves as a competitive dual antagonist against endothelin-1 (ET) by targeting both ET A and ET B receptors. It exhibits binding affinities with K i values of 4.7 nM for ET A and 95 nM for ET B in human SMC.

Bosentan-d4
Other Forms of Bosentan-d4:
Bosentan (hydrate)T6265157212-55-0
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BosentanT6264147536-97-8
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Bosentan-d4

Catalog No. T73820Cas No. 1065472-77-6
Bosentan-d4, the deuterium-labeled variant of Bosentan, serves as a competitive dual antagonist against endothelin-1 (ET) by targeting both ET A and ET B receptors. It exhibits binding affinities with K i values of 4.7 nM for ET A and 95 nM for ET B in human SMC.
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5 mg$68835 days
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Product Introduction

Bioactivity
Description
Bosentan-d4, the deuterium-labeled variant of Bosentan, serves as a competitive dual antagonist against endothelin-1 (ET) by targeting both ET A and ET B receptors. It exhibits binding affinities with K i values of 4.7 nM for ET A and 95 nM for ET B in human SMC.
Chemical Properties
Molecular Weight555.64
FormulaC27H25D4N5O6S
Cas No.1065472-77-6
Storage & Solubility Information
StorageShipping with blue ice.

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