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CB2R-IN-1

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Catalog No. T10697Cas No. 1257555-79-5

CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).

CB2R-IN-1

CB2R-IN-1

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Catalog No. T10697Cas No. 1257555-79-5
CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).
Pack SizePriceAvailabilityQuantity
25 mg1.871 €8-10 weeks
50 mg2.451 €8-10 weeks
100 mg3.230 €8-10 weeks
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Product Introduction

Bioactivity
Description
CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).
Targets&IC50
CB2:0.9 nM (ki)
In vitro
CB2R-IN-1 (Compound 37) exhibits excellent selectivity for the cannabinoid CB2 receptor ligand over the CB1 receptor (Ki: 8259.3 nM).
Chemical Properties
Molecular Weight608.67
FormulaC23H27F3N4O6S3
Cas No.1257555-79-5
Relative Density.1.52 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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Keywords

CB2R-IN-1CB-2R-IN-1CB2RIN1CB2R IN 1
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