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CBK289001

Name: CBK289001
Brand: TargetMol
SKU: T38598
Price: 35 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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Catalog No. T38598Cas No. 1212663-24-5

CBK289001 is a tartrate-resistant acid phosphatase (TRAP/ACP5) inhibitor that inhibits TRAP 5b MV, TRAP 5b OX, and TRAP 5a OX with IC50 values of 125 μM, 4.21 μM, and 14.2 μM, respectively.

CBK289001

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Catalog No. T38598Cas No. 1212663-24-5

CBK289001 is a tartrate-resistant acid phosphatase (TRAP/ACP5) inhibitor that inhibits TRAP 5b MV, TRAP 5b OX, and TRAP 5a OX with IC50 values of 125 μM, 4.21 μM, and 14.2 μM, respectively.

Pack Size	Price	Availability	Quantity
5 mg	$2,389	6-8 weeks

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Product Introduction

Bioactivity

Description	CBK289001 is a tartrate-resistant acid phosphatase (TRAP/ACP5) inhibitor that inhibits TRAP 5b MV, TRAP 5b OX, and TRAP 5a OX with IC50 values of 125 μM, 4.21 μM, and 14.2 μM, respectively.
In vitro	CBK289001 exclusively impedes TRAP3-mediated high cell migration in a dose-dependent manner, demonstrating significant migration inhibition starting 24 hours post-treatment and achieving reduced migration velocity over 30 hours at concentrations of 20 μM or 100 μM. This indicates CBK289001 effectively hinders TRAP-dependent migration in TRAP-overexpressing MDA-MB-231 breast cancer cells.

Chemical Properties

Molecular Weight	396.4
Formula	C₁₉H₂₀N₆O₄
Cas No.	1212663-24-5

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

CBK-289001CBK 289001CBK289001