Shopping Cart
- Remove All
![TargetMol](https://www.targetmol.com/storage/error/oops.webp)
Your shopping cart is currently empty
Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | $446 | 6-8 weeks | |
25 mg | $1,430 | 6-8 weeks | |
50 mg | $1,860 | 6-8 weeks | |
100 mg | $2,500 | 6-8 weeks |
Description | CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM). |
Targets&IC50 | Gastrin/CCK-B:0.43 nM , Gastrin/CCK-A:1.82 μM |
In vivo | CCK-B Receptor Antagonist 2 (0.1 μmol/kg; i.v.) inhibits pentagastrin-induced gastric acid secretion in anesthetized rats, with an ED50 of 8.3 nmol/kg. |
Molecular Weight | 484.55 |
Formula | C27H28N6O3 |
Cas No. | 155412-88-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 250 mg/mL (515.94 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
|
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.