Shopping Cart

Remove All
Your shopping cart is currently empty

Aptiganel hydrochloride

Name: Aptiganel hydrochloride
Brand: TargetMol
SKU: T38068
Price: 197 EUR
Availability: InStock
Rating: 4.5 (1 reviews)

😃Good

Catalog No. T38068Cas No. 137160-11-3

Potent and noncompetitive NMDA receptor antagonist (IC50 = 36 nM). Exhibits >70-fold selectivity for NMDA receptor over σ receptor. Neuroprotective in a rat model of focal ischemia.

Aptiganel hydrochloride

😃Good

Catalog No. T38068Cas No. 137160-11-3

Potent and noncompetitive NMDA receptor antagonist (IC50 = 36 nM). Exhibits >70-fold selectivity for NMDA receptor over σ receptor. Neuroprotective in a rat model of focal ischemia.

Pack Size	Price	Availability	Quantity
2 mg	77 €	5 days

Bulk & Custom

Add to Cart

Questions

Resource Download

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity

Description

Potent and noncompetitive NMDA receptor antagonist (IC50 = 36 nM). Exhibits >70-fold selectivity for NMDA receptor over σ receptor. Neuroprotective in a rat model of focal ischemia.

Chemical Properties

Molecular Weight	339.87
Formula	C₂₀H₂₂ClN₃
Cas No.	137160-11-3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 100 mM

H2O: 50 mM

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	2.9423 mL	14.7115 mL	29.4230 mL	147.1151 mL
5 mM	0.5885 mL	2.9423 mL	5.8846 mL	29.4230 mL
10 mM	0.2942 mL	1.4712 mL	2.9423 mL	14.7115 mL
20 mM	0.1471 mL	0.7356 mL	1.4712 mL	7.3558 mL
50 mM	0.0588 mL	0.2942 mL	0.5885 mL	2.9423 mL

DMSO

	1mg	5mg	10mg	50mg
100 mM	0.0294 mL	0.1471 mL	0.2942 mL	1.4712 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Aptiganel hydrochlorideAptiganel Hydrochloride