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Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $1,520 | 10-14 weeks | |
50 mg | $1,980 | 10-14 weeks | |
100 mg | $2,500 | 10-14 weeks |
Description | CK2 inhibitor 3 is a highly potent inhibitor of protein kinase CK2, exhibiting an IC50 value of 280 nM. It effectively inhibits the intracellular activity of CK2 and displays a notable impact on the viability of tumor cells. Moreover, CK2 inhibitor 3 demonstrates exceptional selectivity among a diverse panel of 320 kinases [1]. |
In vitro | CK2 inhibitor 3 (compound 4) significantly reduces cell viability in Jurkat cells in a dose-dependent manner, with a DC50 value of 12.80 μM after 24 hours at concentrations from 0 to 50 μM [1]. Additionally, at 5 μM and 20 μM over 16 hours, it reduces CK2-dependent phospho-site Akt Ser129 levels, demonstrating targeted efficacy [1]. |
Molecular Weight | 381.2 |
Formula | C13H9BrN4O3S |
Cas No. |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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