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CST 905

CST 905
CST 905, a selective and potent BRAFV600EDegrader (PROTAC) with a DC50 of 18 nM, features a von Hippel Lindau (VHL) E3 ligase ligand connected via a linker to a PLX-derived ligand. Distinctively, CST 905 does not activate ERK, setting it apart from other BRAFV600EDegraders.
Catalog No. T83933
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CST 905

Catalog No. T83933
CST 905, a selective and potent BRAFV600EDegrader (PROTAC) with a DC50 of 18 nM, features a von Hippel Lindau (VHL) E3 ligase ligand connected via a linker to a PLX-derived ligand. Distinctively, CST 905 does not activate ERK, setting it apart from other BRAFV600EDegraders.
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Product Introduction

Bioactivity
Description
CST 905, a selective and potent BRAFV600EDegrader (PROTAC) with a DC50 of 18 nM, features a von Hippel Lindau (VHL) E3 ligase ligand connected via a linker to a PLX-derived ligand. Distinctively, CST 905 does not activate ERK, setting it apart from other BRAFV600EDegraders.
Chemical Properties
Molecular Weight1025.20
FormulaC51H58F2N10O7S2
Cas No.
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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