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Desmethyl Bosentan

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Catalog No. T37351Cas No. 253688-61-8

Desmethyl bosentan, an active metabolite of the endothelin receptor antagonist bosentan, activates the pregnane X receptor (PXR) in CV-1 monkey kidney cells expressing the human receptor in a reporter assay at a concentration of 25 μM.

Desmethyl Bosentan

Desmethyl Bosentan

😃Good
Catalog No. T37351Cas No. 253688-61-8
Desmethyl bosentan, an active metabolite of the endothelin receptor antagonist bosentan, activates the pregnane X receptor (PXR) in CV-1 monkey kidney cells expressing the human receptor in a reporter assay at a concentration of 25 μM.
Pack SizePriceAvailabilityQuantity
500 μg$29635 days
1 mg$54535 days
5 mg$2,40035 days
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Product Introduction

Bioactivity
Description
Desmethyl bosentan, an active metabolite of the endothelin receptor antagonist bosentan, activates the pregnane X receptor (PXR) in CV-1 monkey kidney cells expressing the human receptor in a reporter assay at a concentration of 25 μM.
Chemical Properties
Molecular Weight537.59
FormulaC26H27N5O6S
Cas No.253688-61-8
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: Soluble
Acetonitrile: Soluble
Methanol: Soluble

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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Desmethyl Bosentan
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