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DRAK2-IN-1

Catalog No. T11094Cas No. 871837-60-4

Drak2-in-1, a potent, selective and ATP-competitive DRAK2 inhibitor, has an IC50 and KIvalue of 3 nM and 0.26 nM, respectively.Drak2-in-1 also had an effect on DRAK1 (IC50=51 nM).

DRAK2-IN-1

DRAK2-IN-1

Catalog No. T11094Cas No. 871837-60-4
Drak2-in-1, a potent, selective and ATP-competitive DRAK2 inhibitor, has an IC50 and KIvalue of 3 nM and 0.26 nM, respectively.Drak2-in-1 also had an effect on DRAK1 (IC50=51 nM).
Pack SizePriceAvailabilityQuantity
25 mg$7666-8 weeks
50 mg$9956-8 weeks
100 mg$1,7406-8 weeks
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Product Introduction

Bioactivity
Description
Drak2-in-1, a potent, selective and ATP-competitive DRAK2 inhibitor, has an IC50 and KIvalue of 3 nM and 0.26 nM, respectively.Drak2-in-1 also had an effect on DRAK1 (IC50=51 nM).
Targets&IC50
DRPK2:1.8 μM , DRAK1:51 nM , DRAK2:2.3 μM , DRAK2:3 nM , DRPK3:1.8 μM
Chemical Properties
Molecular Weight376.41
FormulaC21H20N4O3
Cas No.871837-60-4
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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Keywords

DRAK2IN1DRAK2 IN 1DRAK2-IN-1DRAK-2-IN-1
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