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EGFR-IN-52

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Catalog No. T61646Cas No. 454436-75-0

EGFR-IN-52 (Compound 4) is a highly effective inhibitor of the epidermal growth factor receptor (EGFR) with IC50 values of 0.358, 86.02, and 432.67 μM against EGFR, EGFR L858R-TK, and EGFR T790M-TK, respectively. Additionally, it demonstrates potent cytotoxic effects on cancer cell lines and triggers apoptosis [1].

EGFR-IN-52

EGFR-IN-52

😃Good
Catalog No. T61646Cas No. 454436-75-0
EGFR-IN-52 (Compound 4) is a highly effective inhibitor of the epidermal growth factor receptor (EGFR) with IC50 values of 0.358, 86.02, and 432.67 μM against EGFR, EGFR L858R-TK, and EGFR T790M-TK, respectively. Additionally, it demonstrates potent cytotoxic effects on cancer cell lines and triggers apoptosis [1].
Pack SizePriceAvailabilityQuantity
25 mg$2,1406-8 weeks
50 mg$2,7856-8 weeks
100 mg$3,5206-8 weeks
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Product Introduction

Bioactivity
Description
EGFR-IN-52 (Compound 4) is a highly effective inhibitor of the epidermal growth factor receptor (EGFR) with IC50 values of 0.358, 86.02, and 432.67 μM against EGFR, EGFR L858R-TK, and EGFR T790M-TK, respectively. Additionally, it demonstrates potent cytotoxic effects on cancer cell lines and triggers apoptosis [1].
Chemical Properties
Molecular Weight382.44
FormulaC19H18N4O3S
Cas No.454436-75-0
Storage & Solubility Information
StorageShipping with blue ice.

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