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Emedastine Difumarate
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Catalog No. T21388Cas No. 87233-62-3
Alias Rapimine, KB-2413, KB 2413, Emedastine fumarate, DSSTox_CID_26911, AL-3432A
Emedastine Difumarate is a selective histamine H1 receptor antagonist with anti-allergic activity, prescribed for allergic conjunctivitis. Upon ocular administration, emedastine causes a dose-dependent inhibition of histamine-stimulated vascular permeability in the conjunctiva.
Emedastine Difumarate
😃Good
Catalog No. T21388Alias Rapimine, KB-2413, KB 2413, Emedastine fumarate, DSSTox_CID_26911, AL-3432ACas No. 87233-62-3
Emedastine Difumarate is a selective histamine H1 receptor antagonist with anti-allergic activity, prescribed for allergic conjunctivitis. Upon ocular administration, emedastine causes a dose-dependent inhibition of histamine-stimulated vascular permeability in the conjunctiva.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $970 | 7-10 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Emedastine Difumarate is a selective histamine H1 receptor antagonist with anti-allergic activity, prescribed for allergic conjunctivitis. Upon ocular administration, emedastine causes a dose-dependent inhibition of histamine-stimulated vascular permeabil |
| Targets&IC50 | H1 receptor:1.3 nM (Ki), H3 receptor:12430 nM (Ki), H2 receptor:49067 nM (Ki) |
| Alias | Rapimine, KB-2413, KB 2413, Emedastine fumarate, DSSTox_CID_26911, AL-3432A |
| Molecular Weight | 534.56 |
| Formula | C25H34N4O9 |
| Cas No. | 87233-62-3 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | H2O: Insoluble DMSO: Soluble |
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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