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EPI-7170

Catalog No. T63811Cas No. 2139288-26-7

EPI-7170 is a ralaniten analogue and a potent antagonist of the androgen receptor N-terminal structural domain, blocking the transcriptional activity of the full-length AR (FL-AR) and AR splice variants (AR-Vs). EPI-7170 exhibits antitumor activity against enzalutamide resistant debulking resistant prostate cancer (CRPC).

EPI-7170

EPI-7170

Catalog No. T63811Cas No. 2139288-26-7
EPI-7170 is a ralaniten analogue and a potent antagonist of the androgen receptor N-terminal structural domain, blocking the transcriptional activity of the full-length AR (FL-AR) and AR splice variants (AR-Vs). EPI-7170 exhibits antitumor activity against enzalutamide resistant debulking resistant prostate cancer (CRPC).
Pack SizePriceAvailabilityQuantity
25 mg$9318-10 weeks
50 mg$1,2108-10 weeks
100 mg$1,9408-10 weeks
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Product Introduction

Bioactivity
Description
EPI-7170 is a ralaniten analogue and a potent antagonist of the androgen receptor N-terminal structural domain, blocking the transcriptional activity of the full-length AR (FL-AR) and AR splice variants (AR-Vs). EPI-7170 exhibits antitumor activity against enzalutamide resistant debulking resistant prostate cancer (CRPC).
Chemical Properties
Molecular Weight540.88
FormulaC22H28Cl3NO6S
Cas No.2139288-26-7
Storage & Solubility Information
StorageShipping with blue ice.

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