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EST64454 Maleic acid salt

Name: EST64454 Maleic acid salt
Brand: TargetMol
SKU: T9306
Price: 80 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T9306Cas No. 2088272-67-5

EST64454 Maleic acid salt is the maleic acid salt form of EST64454.EST64454 is a highly soluble σ1 receptor antagonist clinical candidate for the treatment of pain.

EST64454 Maleic acid salt

🥰Excellent

Purity: 97.54%

Catalog No. T9306Cas No. 2088272-67-5

EST64454 Maleic acid salt is the maleic acid salt form of EST64454.EST64454 is a highly soluble σ1 receptor antagonist clinical candidate for the treatment of pain.

Pack Size	Price	Availability
1 mg	$80	In Stock
5 mg	$181	In Stock
10 mg	$272	In Stock
25 mg	$448	In Stock
50 mg	$630	In Stock
100 mg	$852	In Stock
200 mg	$1,130	In Stock
1 mL x 10 mM (in DMSO)	$218	In Stock

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Purity:97.54%

Resource Download

COA LCMS HNMR HPLC

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Product Introduction

Bioactivity

Description

EST64454 Maleic acid salt is the maleic acid salt form of EST64454.EST64454 is a highly soluble σ1 receptor antagonist clinical candidate for the treatment of pain.

Chemical Properties

Molecular Weight	480.46
Formula	C₂₂H₂₆F₂N₄O₆
Cas No.	2088272-67-5
Smiles	CC(N1CCN(CCOCC2=NN(C3=CC=C(F)C(F)=C3)C=C2)CC1)=O.O=C(O)/C=C\C(O)=O
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 60 mg/ml (124.88 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0813 mL	10.4067 mL	20.8134 mL	104.0669 mL
5 mM	0.4163 mL	2.0813 mL	4.1627 mL	20.8134 mL
10 mM	0.2081 mL	1.0407 mL	2.0813 mL	10.4067 mL
20 mM	0.1041 mL	0.5203 mL	1.0407 mL	5.2033 mL
50 mM	0.0416 mL	0.2081 mL	0.4163 mL	2.0813 mL
100 mM	0.0208 mL	0.1041 mL	0.2081 mL	1.0407 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

EST-64454 Maleic acid saltEST64454 Maleic acid saltEST64454 Maleic acid