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Etifoxine

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Etifoxine

Catalog No. T13691Cas No. 21715-46-8

Etifoxine preferentially acts on β2 or β3 subunit-containing GABAA receptors. GABAA receptor Etifoxine exhibits anxiolytic activity in rodents and humans with no sedative, myorelaxant or mnesic side effects. Etifoxine acts as a ligand of the translocator protein (TSPO); promotes axonal regeneration. Etifoxine(HOE 36-801) is potentiator of GABAA receptor function in cultured neurons.

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Pack Size	Price	Availability	Quantity
2 mg	$35	5 days

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Product Introduction

Bioactivity

Description	Etifoxine preferentially acts on β2 or β3 subunit-containing GABAA receptors. GABAA receptor Etifoxine exhibits anxiolytic activity in rodents and humans with no sedative, myorelaxant or mnesic side effects. Etifoxine acts as a ligand of the translocator protein (TSPO); promotes axonal regeneration. Etifoxine(HOE 36-801) is potentiator of GABAA receptor function in cultured neurons.
Alias	HOE 36-801

Chemical Properties

Molecular Weight	300.78
Formula	C17H17ClN2O
Cas No.	21715-46-8

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 100 mg/mL (332.47 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.3247 mL	16.6234 mL	33.2469 mL	166.2345 mL
5 mM	0.6649 mL	3.3247 mL	6.6494 mL	33.2469 mL
10 mM	0.3325 mL	1.6623 mL	3.3247 mL	16.6234 mL
20 mM	0.1662 mL	0.8312 mL	1.6623 mL	8.3117 mL
50 mM	0.0665 mL	0.3325 mL	0.6649 mL	3.3247 mL
100 mM	0.0332 mL	0.1662 mL	0.3325 mL	1.6623 mL

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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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Keywords

Etifoxine