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Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $1,970 | 8-10 weeks | |
50 mg | $2,580 | 8-10 weeks | |
100 mg | $3,400 | 8-10 weeks |
Description | Frakefamide is a potent analgesic that functions as a peripheral active μ-selective receptor agonist. It cannot penetrate the blood-brain barrier to enter the central nervous system. |
In vivo | Frakefamide exhibits a dose-dependent enhancement in morphine-appropriate responses, reaching 50% at the maximal tested dose (10 μmol/kg) following a 2-minute infusion period. However, after 15-minute infusions, the peak morphine-appropriate response achieved is 25% at a dose of 17.5 μmol/kg [1,2]. |
Molecular Weight | 563.62 |
Formula | C30H34FN5O5 |
Cas No. | 188196-22-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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