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Pack Size | Price | Availability | Quantity |
---|---|---|---|
100 mg | $1,110 | 10-14 weeks | |
200 mg | $1,690 | 10-14 weeks |
Description | GAK inhibitor 49 hydrochloride is a potent, ATP-competitive and highly selective inhibitor of cyclin G associated kinase (GAK) with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 hydrochloride can also bind to RIPK2. |
In vitro | GAK inhibitor 49 (compound 49) hydrochloride demonstrates limited inhibition towards AAK1, BMP2K, and STK16, exhibiting IC50 values of 28, 63, and >100μM, respectively [1]. |
Molecular Weight | 406.86 |
Formula | C20H23ClN2O5 |
Cas No. |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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