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Glucagon receptor antagonists-5

Name: Glucagon receptor antagonists-5
Brand: TargetMol
SKU: T11416
Price: 28 EUR
Availability: InStock
Rating: 4.5 (1 reviews)

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Catalog No. T11416Cas No. 2200274-63-9

Glucagon receptor antagonists-5 is an orally bioavailable indazole-based glucagon receptor antagonist (Ki: 32 nM). It has potential for the treatment of type 2 diabetes mellitus (T2DM).

Glucagon receptor antagonists-5

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Catalog No. T11416Cas No. 2200274-63-9

Glucagon receptor antagonists-5 is an orally bioavailable indazole-based glucagon receptor antagonist (Ki: 32 nM). It has potential for the treatment of type 2 diabetes mellitus (T2DM).

Pack Size	Price	Availability
25 mg	$1,520	6-8 weeks
50 mg	$1,980	6-8 weeks
100 mg	$2,500	6-8 weeks

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Product Introduction

Bioactivity

Description	Glucagon receptor antagonists-5 is an orally bioavailable indazole-based glucagon receptor antagonist (Ki: 32 nM). It has potential for the treatment of type 2 diabetes mellitus (T2DM).
Targets&IC50	Glucagon receptor:ki:32 nM

Chemical Properties

Molecular Weight	572.02
Formula	C₃₀H₂₉ClF₃N₃O₃
Cas No.	2200274-63-9
Relative Density.	1.31 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

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Keywords

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