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GRK2 Inhibitor 2

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Catalog No. T79913Cas No. 2592436-21-8

GRK2 Inhibitor 2 (Compound 8h), with an IC50 of 19 nM for GRK2 and 137 nM for Aurora-A, enhances β-AR-mediated cAMP accumulation in GRK2-overexpressing HEK293 cells. It is utilized in congestive heart failure (HF) research [1].

GRK2 Inhibitor 2

GRK2 Inhibitor 2

😃Good
Catalog No. T79913Cas No. 2592436-21-8
GRK2 Inhibitor 2 (Compound 8h), with an IC50 of 19 nM for GRK2 and 137 nM for Aurora-A, enhances β-AR-mediated cAMP accumulation in GRK2-overexpressing HEK293 cells. It is utilized in congestive heart failure (HF) research [1].
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50 mgInquiry8-10 weeks
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Product Introduction

Bioactivity
Description
GRK2 Inhibitor 2 (Compound 8h), with an IC50 of 19 nM for GRK2 and 137 nM for Aurora-A, enhances β-AR-mediated cAMP accumulation in GRK2-overexpressing HEK293 cells. It is utilized in congestive heart failure (HF) research [1].
Chemical Properties
Molecular Weight332.36
FormulaC19H16N4O2
Cas No.2592436-21-8
Storage & Solubility Information
StorageShipping with blue ice.

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