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GRK5-IN-3

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Catalog No. T62599Cas No. 2410793-22-3

GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), significantly inhibiting GRK5 with an IC50 of 0.22 μM and GRK6 with an IC50 of 0.41 μM.

GRK5-IN-3

GRK5-IN-3

😃Good
Catalog No. T62599Cas No. 2410793-22-3
GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), significantly inhibiting GRK5 with an IC50 of 0.22 μM and GRK6 with an IC50 of 0.41 μM.
Pack SizePriceAvailabilityQuantity
25 mg$1,5206-8 weeks
50 mg$1,9806-8 weeks
100 mg$2,5006-8 weeks
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Product Introduction

Bioactivity
Description
GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), significantly inhibiting GRK5 with an IC50 of 0.22 μM and GRK6 with an IC50 of 0.41 μM.
Chemical Properties
Molecular Weight443.46
FormulaC23H21N7O3
Cas No.2410793-22-3
Storage & Solubility Information
StorageShipping with blue ice.

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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