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GSK097 is a highly potent and selective inhibitor of the second bromodomain (BD2) found in bromodomain and extra-terminal domain (BET) proteins. It exhibits a remarkable 2000-fold selectivity for BD2 over BD1, as indicated by BRD4 data. Additionally, GSK097 demonstrates solubility of over 1 mg/mL in FaSSIF media.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | 921 € | Backorder |
Description | GSK097 is a highly potent and selective inhibitor of the second bromodomain (BD2) found in bromodomain and extra-terminal domain (BET) proteins. It exhibits a remarkable 2000-fold selectivity for BD2 over BD1, as indicated by BRD4 data. Additionally, GSK097 demonstrates solubility of over 1 mg/mL in FaSSIF media. |
In vitro | GSK097 exhibits potent inhibitory activity, as indicated by pIC50 values of 7.4, 8.0, 7.6, and 7.9, against BRD2 (BD2), BRD3 (BD2), BRD4 (BD2), and BRDT (BD2), respectively[1]. |
Molecular Weight | 339.395 |
Formula | C19H21N3O3 |
Cas No. | 2159137-02-5 |
Relative Density. | 1.29 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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