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LY487379

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Catalog No. T62756Cas No. 353231-17-1

LY487379 is a selective human mGluR2 positive allosteric modulator (PAM) that enhances glutamate-stimulated [35 S] GTPγS binding to mGlu2 receptors (EC50: 1.7 μM) and mGlu3 receptors (EC50 >10 μM). LY487379 induces cognitive flexibility and behavioral inhibition in a rat model and can be used to study schizophrenia.

LY487379
Other Forms of LY487379:
LY487379 hydrochlorideT22955353229-59-1
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LY487379

😃Good
Catalog No. T62756Cas No. 353231-17-1
LY487379 is a selective human mGluR2 positive allosteric modulator (PAM) that enhances glutamate-stimulated [35 S] GTPγS binding to mGlu2 receptors (EC50: 1.7 μM) and mGlu3 receptors (EC50 >10 μM). LY487379 induces cognitive flexibility and behavioral inhibition in a rat model and can be used to study schizophrenia.
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2 mg38 €5 days
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Product Introduction

Bioactivity
Description
LY487379 is a selective human mGluR2 positive allosteric modulator (PAM) that enhances glutamate-stimulated [35 S] GTPγS binding to mGlu2 receptors (EC50: 1.7 μM) and mGlu3 receptors (EC50 >10 μM). LY487379 induces cognitive flexibility and behavioral inhibition in a rat model and can be used to study schizophrenia.
Chemical Properties
Molecular Weight452.45
FormulaC21H19F3N2O4S
Cas No.353231-17-1
Storage & Solubility Information
StorageShipping with blue ice.

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