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MA242 free base

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Catalog No. T62977Cas No. 1049704-17-7

MA242 free base is a specific dual inhibitor of MDM2 and NFAT1 that induces apoptosis in pancreatic cancer cell lines. It binds directly to MDM2 and NFAT1 with high affinity, induces their protein degradation, and inhibits NFAT1-mediated MDM2 transcription.

MA242 free base
Other Forms of MA242 free base:
MA242T119311049704-18-8
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MA242 free base

😃Good
Catalog No. T62977Cas No. 1049704-17-7
MA242 free base is a specific dual inhibitor of MDM2 and NFAT1 that induces apoptosis in pancreatic cancer cell lines. It binds directly to MDM2 and NFAT1 with high affinity, induces their protein degradation, and inhibits NFAT1-mediated MDM2 transcription.
Pack SizePriceAvailabilityQuantity
25 mg$2,14010-14 weeks
50 mg$2,78510-14 weeks
100 mg$3,52010-14 weeks
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Product Introduction

Bioactivity
Description
MA242 free base is a specific dual inhibitor of MDM2 and NFAT1 that induces apoptosis in pancreatic cancer cell lines. It binds directly to MDM2 and NFAT1 with high affinity, induces their protein degradation, and inhibits NFAT1-mediated MDM2 transcription.
Chemical Properties
Molecular Weight465.95
FormulaC24H20ClN3O3S
Cas No.1049704-17-7
Storage & Solubility Information
StorageShipping with blue ice.

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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