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MrgprX2 antagonist-4

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Catalog No. T40268Cas No. 2641398-04-9
Alias MrgprX2 antagonist-4

MrgprX2 antagonist-4 and compound B-51 E117, is a potent MrgprX2 antagonist. It specifically targets and inhibits the MrgprX2 receptor, making it suitable for investigating various inflammatory skin disorders.

MrgprX2 antagonist-4

MrgprX2 antagonist-4

😃Good
Catalog No. T40268Alias MrgprX2 antagonist-4Cas No. 2641398-04-9
MrgprX2 antagonist-4 and compound B-51 E117, is a potent MrgprX2 antagonist. It specifically targets and inhibits the MrgprX2 receptor, making it suitable for investigating various inflammatory skin disorders.
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Product Introduction

Bioactivity
Description
MrgprX2 antagonist-4 and compound B-51 E117, is a potent MrgprX2 antagonist. It specifically targets and inhibits the MrgprX2 receptor, making it suitable for investigating various inflammatory skin disorders.
In vitro
MRGPRX2, a member of the Mas-related gene family, is expressed in sensory neurons, mast cells, and keratinocytes. MRGPRX2 mRNA is present in adipose tissue, esophagus, urinary bladder, and lungs, with the highest levels in skin. Activation of MRGPRX2 results in mast cell degranulation and subsequent pseudo-allergic reactions[2].
AliasMrgprX2 antagonist-4
Chemical Properties
Molecular Weight269.348
FormulaC16H19N3O
Cas No.2641398-04-9
Relative Density.1.23 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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