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PARP/EZH2-IN-1

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Catalog No. T40310Cas No. 2687273-52-3
Alias PARP/EZH2-IN-1

PARP/EZH2-IN-1 is a novel dual inhibitor targeting PARP (IC50 6.87 nM) and EZH2 (IC50 36.51 nM), showing promising potential for treating triple-negative breast cancer with wild-type BRCA.

PARP/EZH2-IN-1

PARP/EZH2-IN-1

😃Good
Catalog No. T40310Alias PARP/EZH2-IN-1Cas No. 2687273-52-3
PARP/EZH2-IN-1 is a novel dual inhibitor targeting PARP (IC50 6.87 nM) and EZH2 (IC50 36.51 nM), showing promising potential for treating triple-negative breast cancer with wild-type BRCA.
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5 mg$970Backorder
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Product Introduction

Bioactivity
Description
PARP/EZH2-IN-1 is a novel dual inhibitor targeting PARP (IC50 6.87 nM) and EZH2 (IC50 36.51 nM), showing promising potential for treating triple-negative breast cancer with wild-type BRCA.
Targets&IC50
PARP1:6.87 nM (IC50), EZH2:36.51 nM (IC50)
AliasPARP/EZH2-IN-1
Chemical Properties
Molecular Weight768.85
FormulaC43H41FN8O5
Cas No.2687273-52-3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Keywords

PARP/EZH2 IN 1PARP/EZH-2-IN-1PARP/EZH2IN1
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