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PD-159020

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Catalog No. T12382Cas No. 177904-00-6

PD-159020 is a non-selective antagonist of ETA/ETB (hETA and hETB) with IC50 values of 30 nM and 50 nM, respectively.

PD-159020

PD-159020

😃Good
Catalog No. T12382Cas No. 177904-00-6
PD-159020 is a non-selective antagonist of ETA/ETB (hETA and hETB) with IC50 values of 30 nM and 50 nM, respectively.
Pack SizePriceAvailabilityQuantity
25 mg$1,5206-8 weeks
50 mg$1,9806-8 weeks
100 mg$2,5006-8 weeks
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Product Introduction

Bioactivity
Description
PD-159020 is a non-selective antagonist of ETA/ETB (hETA and hETB) with IC50 values of 30 nM and 50 nM, respectively.
Targets&IC50
ETB (human):50 nM , ETA (human):30 nM
In vitro
PD-159020 exhibits potent inhibitory activity against arachidonic acid release, AAR-B, with an IC50 of 0.23 μM.
Chemical Properties
Molecular Weight551.54
FormulaC32H25NO8
Cas No.177904-00-6
Relative Density.1.41 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Keywords

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