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PDGFR-IN-1

🥰Excellent
Catalog No. T62872Cas No. 2644673-07-2

PDGFR-IN-1 (compound 7m) is an orally active PDGFR (platelet-derived growth factor receptor) inhibitor that targets PDGFRα (IC50: 2.4 nM) and PDGFRβ (IC50: 0.9 nM), exhibiting strong anti-tumor effects and low toxicity, making it suitable for osteosarcoma studies.

PDGFR-IN-1

PDGFR-IN-1

🥰Excellent
Catalog No. T62872Cas No. 2644673-07-2
PDGFR-IN-1 (compound 7m) is an orally active PDGFR (platelet-derived growth factor receptor) inhibitor that targets PDGFRα (IC50: 2.4 nM) and PDGFRβ (IC50: 0.9 nM), exhibiting strong anti-tumor effects and low toxicity, making it suitable for osteosarcoma studies.
Pack SizePriceAvailabilityQuantity
25 mg$1,520In Stock
50 mg$1,980In Stock
100 mg$2,500In Stock
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Product Introduction

Bioactivity
Description
PDGFR-IN-1 (compound 7m) is an orally active PDGFR (platelet-derived growth factor receptor) inhibitor that targets PDGFRα (IC50: 2.4 nM) and PDGFRβ (IC50: 0.9 nM), exhibiting strong anti-tumor effects and low toxicity, making it suitable for osteosarcoma studies.
Chemical Properties
Molecular Weight458.56
FormulaC25H30N8O
Cas No.2644673-07-2
SmilesO(C)C1=C(C=CC(NC=2N=C(NC=3C=C4C(=CC3)C=NN4)C(C)=CN2)=C1)N5CCN(CC)CC5
Storage & Solubility Information
Storagekeep away from moisture,store at low temperature | Shipping with blue ice.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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