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PLK1/BRD4-IN-2

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Catalog No. T87220Cas No. 2251709-89-2

PLK1/BRD4-IN-2 (compound 15), an analog of BI-2536, simultaneously inhibits both Polo-like kinase 1 (PLK1 IC 50 = 40 nM) and BRD4 bromodomain (BRD4-BD1 IC 50 = 28 nM) as a dual inhibitor [1].

PLK1/BRD4-IN-2

PLK1/BRD4-IN-2

😃Good
Catalog No. T87220Cas No. 2251709-89-2
PLK1/BRD4-IN-2 (compound 15), an analog of BI-2536, simultaneously inhibits both Polo-like kinase 1 (PLK1 IC 50 = 40 nM) and BRD4 bromodomain (BRD4-BD1 IC 50 = 28 nM) as a dual inhibitor [1].
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50 mgInquiry10-14 weeks
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Product Introduction

Bioactivity
Description
PLK1/BRD4-IN-2 (compound 15), an analog of BI-2536, simultaneously inhibits both Polo-like kinase 1 (PLK1 IC 50 = 40 nM) and BRD4 bromodomain (BRD4-BD1 IC 50 = 28 nM) as a dual inhibitor [1].
Chemical Properties
Molecular Weight492.61
FormulaC27H36N6O3
Cas No.2251709-89-2
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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