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Ruboxistaurin mesylate monohydrate

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Catalog No. T69990Cas No. 202260-21-7

Ruboxistaurin mesylate monohydrate is a PKC beta inhibitor potentially for the treatment of diabetic nephropathy and diabetic macular edema. Ruboxistaurin attenuates diabetic nephropathy via modulation of TGF-β1/Smad and GRAP pathways. Ruboxistaurin reduces oxidative stress and attenuates left ventricular hypertrophy and dysfunction in rats with streptozotocin-induced diabetes. Ruboxistaurin inhibits retinal neovascularization via suppression of phosphorylation of ERK1/2 and Akt.

Ruboxistaurin mesylate monohydrate
Other Forms of Ruboxistaurin mesylate monohydrate:

Ruboxistaurin mesylate monohydrate

😃Good
Catalog No. T69990Cas No. 202260-21-7
Ruboxistaurin mesylate monohydrate is a PKC beta inhibitor potentially for the treatment of diabetic nephropathy and diabetic macular edema. Ruboxistaurin attenuates diabetic nephropathy via modulation of TGF-β1/Smad and GRAP pathways. Ruboxistaurin reduces oxidative stress and attenuates left ventricular hypertrophy and dysfunction in rats with streptozotocin-induced diabetes. Ruboxistaurin inhibits retinal neovascularization via suppression of phosphorylation of ERK1/2 and Akt.
Pack SizePriceAvailabilityQuantity
25 mg$2,5701-2 weeks
50 mg$3,3801-2 weeks
100 mg$4,6001-2 weeks
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Product Introduction

Bioactivity
Description
Ruboxistaurin mesylate monohydrate is a PKC beta inhibitor potentially for the treatment of diabetic nephropathy and diabetic macular edema. Ruboxistaurin attenuates diabetic nephropathy via modulation of TGF-β1/Smad and GRAP pathways. Ruboxistaurin reduces oxidative stress and attenuates left ventricular hypertrophy and dysfunction in rats with streptozotocin-induced diabetes. Ruboxistaurin inhibits retinal neovascularization via suppression of phosphorylation of ERK1/2 and Akt.
Chemical Properties
Molecular Weight582.67
FormulaC29H34N4O7S
Cas No.202260-21-7
Storage & Solubility Information
StorageShipping with blue ice.

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Keywords

Ruboxistaurin mesylate MonohydrateDifenamizole hydrochlorideRuboxistaurin Mesylate
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