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SB-612111 hydrochloride

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Catalog No. T62805

SB-612111 hydrochloride is a potent, novel orphan receptor for opioid receptors (ORL-1) antagonist with high affinity for hORL-1 and a Ki value of 0.33 nM. SB-612111 hydrochloride is able to act on mu-receptor (Ki: 57.6 nM), κ SB-612111 hydrochloride effectively antagonized the nociceptive effects of Nociceptin in an acute pain model.

SB-612111 hydrochloride

SB-612111 hydrochloride

😃Good
Catalog No. T62805
SB-612111 hydrochloride is a potent, novel orphan receptor for opioid receptors (ORL-1) antagonist with high affinity for hORL-1 and a Ki value of 0.33 nM. SB-612111 hydrochloride is able to act on mu-receptor (Ki: 57.6 nM), κ SB-612111 hydrochloride effectively antagonized the nociceptive effects of Nociceptin in an acute pain model.
Pack SizePriceAvailabilityQuantity
25 mg$99310-14 weeks
50 mg$1,29010-14 weeks
100 mg$1,99710-14 weeks
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Product Introduction

Bioactivity
Description
SB-612111 hydrochloride is a potent, novel orphan receptor for opioid receptors (ORL-1) antagonist with high affinity for hORL-1 and a Ki value of 0.33 nM. SB-612111 hydrochloride is able to act on mu-receptor (Ki: 57.6 nM), κ SB-612111 hydrochloride effectively antagonized the nociceptive effects of Nociceptin in an acute pain model.
Chemical Properties
Molecular Weight454.86
FormulaC24H30Cl3NO
Storage & Solubility Information
StorageShipping with blue ice.

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