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Selatogrel
🥰Excellent
Catalog No. T71364Cas No. 1159500-34-1
Alias ACT-246475, ACT246475
Selatogrel (ACT-246475) is a selective and potent P2Y12 receptor antagonist with antithrombotic activity and inhibition of platelet aggregation for the study of acute myocardial infarction.
Selatogrel
🥰Excellent
Catalog No. T71364Alias ACT-246475, ACT246475Cas No. 1159500-34-1
Selatogrel (ACT-246475) is a selective and potent P2Y12 receptor antagonist with antithrombotic activity and inhibition of platelet aggregation for the study of acute myocardial infarction.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $457 | In Stock | |
| 5 mg | $1,060 | In Stock | |
| 10 mg | $1,420 | In Stock | |
| 25 mg | $2,120 | In Stock | |
| 50 mg | $2,780 | In Stock |
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Selatogrel (ACT-246475) is a selective and potent P2Y12 receptor antagonist with antithrombotic activity and inhibition of platelet aggregation for the study of acute myocardial infarction. |
| Targets&IC50 | P2Y12 receptor:8 nM |
| In vitro | Selatogrel (ACT-246475) is a reversible and selective P2Y12 receptor antagonist with an IC50 of 8 nM that achieves its effects by inhibiting platelet aggregation. [1] |
| In vivo | Selatogrel (0-0.1 mg/kg, single dose i.v.) inhibits FeCl3-induced thrombosis in wistar rats in a dose-dependent manner and is effective in reducing intraoperative blood loss. [1] |
| Alias | ACT-246475, ACT246475 |
| Molecular Weight | 618.62 |
| Formula | C28H39N6O8P |
| Cas No. | 1159500-34-1 |
| Smiles | C(N[C@H](C(=O)N1CCN(C(OCCCC)=O)CC1)CP(=O)(O)O)(=O)C2=CC(=NC(=N2)C3=CC=CC=C3)N4C[C@@H](OC)CC4 |
Storage & Solubility Information
| Storage | keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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