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SirReal1-O-propargyl, a moiety based on SirReal1, is a selective and highly potent inhibitor of Sirtuin 2 (Sirt2), demonstrating an IC50 of 2.4 μM. It operates by binding to the cereblon ligand through a linker, facilitating the formation of PROTAC for the degradation of Sirt2[1].
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100 mg | Inquiry | Backorder | |
500 mg | Inquiry | Backorder |
Description | SirReal1-O-propargyl, a moiety based on SirReal1, is a selective and highly potent inhibitor of Sirtuin 2 (Sirt2), demonstrating an IC50 of 2.4 μM. It operates by binding to the cereblon ligand through a linker, facilitating the formation of PROTAC for the degradation of Sirt2[1]. |
Targets&IC50 | SIRT2:2.4 μM (IC50) |
Alias | PROTAC Sirt2-binding moiety 1 |
Molecular Weight | 424.54 |
Formula | C21H20N4O2S2 |
Cas No. | 1862237-99-7 |
Relative Density. | 1.34 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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