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TGFβRI-IN-4

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Catalog No. T62559Cas No. 2421135-03-5

TGFβRI-IN-4 is a potent, orally active TGFβ receptor type I kinase (TGFβRI) inhibitor that targets ALK5 (IC50: 44 nM) and NIH3T3 (IC50: 42.5 nM), inhibiting tumor growth and weight in a xenograft tumor model.

TGFβRI-IN-4

TGFβRI-IN-4

😃Good
Catalog No. T62559Cas No. 2421135-03-5
TGFβRI-IN-4 is a potent, orally active TGFβ receptor type I kinase (TGFβRI) inhibitor that targets ALK5 (IC50: 44 nM) and NIH3T3 (IC50: 42.5 nM), inhibiting tumor growth and weight in a xenograft tumor model.
Pack SizePriceAvailabilityQuantity
25 mg$2,1406-8 weeks
50 mg$2,7856-8 weeks
100 mg$3,5206-8 weeks
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Product Introduction

Bioactivity
Description
TGFβRI-IN-4 is a potent, orally active TGFβ receptor type I kinase (TGFβRI) inhibitor that targets ALK5 (IC50: 44 nM) and NIH3T3 (IC50: 42.5 nM), inhibiting tumor growth and weight in a xenograft tumor model.
Chemical Properties
Molecular Weight441.47
FormulaC23H25F2N5O2
Cas No.2421135-03-5
Storage & Solubility Information
StorageShipping with blue ice.

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