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TGFβRI-IN-5

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Catalog No. T60931Cas No. 2541690-15-5

TGFβRI-IN-5 (Compound 4b) is a potent TGFβRI inhibitor with an IC50 of 0.08 μM, demonstrating significant anticancer activity by enhancing apoptosis and arresting the G2/M phase of the cell cycle in all tested cell lines[1].

TGFβRI-IN-5

TGFβRI-IN-5

😃Good
Catalog No. T60931Cas No. 2541690-15-5
TGFβRI-IN-5 (Compound 4b) is a potent TGFβRI inhibitor with an IC50 of 0.08 μM, demonstrating significant anticancer activity by enhancing apoptosis and arresting the G2/M phase of the cell cycle in all tested cell lines[1].
Pack SizePriceAvailabilityQuantity
25 mg$1,5206-8 weeks
50 mg$1,9806-8 weeks
100 mg$2,5006-8 weeks
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Product Introduction

Bioactivity
Description
TGFβRI-IN-5 (Compound 4b) is a potent TGFβRI inhibitor with an IC50 of 0.08 μM, demonstrating significant anticancer activity by enhancing apoptosis and arresting the G2/M phase of the cell cycle in all tested cell lines[1].
Chemical Properties
Molecular Weight328.28
FormulaC16H12N2O6
Cas No.2541690-15-5
Storage & Solubility Information
StorageShipping with blue ice.

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