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[D-Ala2] Leu-Enkephalinamide

Name: [D-Ala2] Leu-Enkephalinamide
Brand: TargetMol
SKU: T83504
Price: 41 EUR
Availability: InStock
Rating: 4.5 (1 reviews)

[D-Ala2] Leu-Enkephalinamide, an enkephalin analog, exhibits significant corneal permeability and analgesic properties, making it suitable for ocular disease research [1] [2].

Catalog No. T83504Cas No. 65189-64-2

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[D-Ala2] Leu-Enkephalinamide

Catalog No. T83504Cas No. 65189-64-2

[D-Ala2] Leu-Enkephalinamide, an enkephalin analog, exhibits significant corneal permeability and analgesic properties, making it suitable for ocular disease research [1] [2].

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Product Introduction

Bioactivity

Description	[D-Ala2] Leu-Enkephalinamide, an enkephalin analog, exhibits significant corneal permeability and analgesic properties, making it suitable for ocular disease research [1] [2].
In vitro	[D-Ala2] Leu-Enkephalinamide (MEA) functions as an agonist at opioid receptors, selectively binding and modulating neurotransmitter release to produce analgesic effects. It mimics endogenous opioid peptides, primarily targeting mu-type receptors crucial for pain regulation in the central nervous system.
In vivo	D-Ala2-Leu-enkephalinamide administered subcutaneously (s.c.) demonstrates increased activity in morphine-dependent animals [2].

Chemical Properties

Molecular Weight	568.66
Formula	C₂₉H₄₀N₆O₆
Cas No.	65189-64-2

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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