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BIIL-260 hydrochloride is a potent, long-acting, orally active antagonist of the leukotriene B4 (LTB4) receptor, exhibiting anti-inflammatory activity with high affinity for the LTB4 receptor on isolated human neutrophil cell membranes (Ki: 1.7 nM).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $916 | 6-8 weeks | |
50 mg | $1,190 | 6-8 weeks | |
100 mg | $1,890 | 6-8 weeks |
Description | BIIL-260 hydrochloride is a potent, long-acting, orally active antagonist of the leukotriene B4 (LTB4) receptor, exhibiting anti-inflammatory activity with high affinity for the LTB4 receptor on isolated human neutrophil cell membranes (Ki: 1.7 nM). |
Targets&IC50 | NOP:4.2 nM (ki), MOP:ki: 1.8 nM , LTB4 receptor 1110:ki: 1.7 nM |
In vitro | BIIL-260 hydrochloride effectively inhibits LTB4-induced intracellular Ca2+ release in human neutrophils (IC50: 0.82 nM). |
Molecular Weight | 503.03 |
Formula | C30H31ClN2O3 |
Cas No. | 192581-24-1 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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