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CGRP antagonist 1

Catalog No. T13453Cas No. 1123757-49-2

CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.

CGRP antagonist 1

CGRP antagonist 1

Purity: 100%
Catalog No. T13453Cas No. 1123757-49-2
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.
Pack SizePriceAvailabilityQuantity
1 mg$342In Stock
5 mg$828In Stock
10 mg$1,150In Stock
25 mg$1,680In Stock
50 mg$2,290In Stock
100 mg$2,970In Stock
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Purity:100%
ee:100%
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Product Introduction

Bioactivity
Description
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.
Targets&IC50
CGRP receptor:35 nM(Ki), CGRP receptor:57 nM
Chemical Properties
Molecular Weight494.54
FormulaC29H26N4O4
Cas No.1123757-49-2
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 60 mg/mL (121.32 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.0221 mL10.1104 mL20.2208 mL101.1041 mL
5 mM0.4044 mL2.0221 mL4.0442 mL20.2208 mL
10 mM0.2022 mL1.0110 mL2.0221 mL10.1104 mL
20 mM0.1011 mL0.5055 mL1.0110 mL5.0552 mL
50 mM0.0404 mL0.2022 mL0.4044 mL2.0221 mL
100 mM0.0202 mL0.1011 mL0.2022 mL1.0110 mL

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