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CRT0066854

Name: CRT0066854
Brand: TargetMol
SKU: T27089
Rating: 4.5 (1 reviews)

😃Good

Catalog No. T27089Cas No. 1438881-19-6

Alias CRT-0066854, CRT0066854, CRT 0066854

CRT-0066854 is a PKCι and PKCζ inhibitor. CRT0066854 was able to restore polarized morphogenesis in the dysplastic H-Ras spheroids.

CRT0066854

😃Good

Catalog No. T27089Alias CRT-0066854, CRT0066854, CRT 0066854Cas No. 1438881-19-6

CRT-0066854 is a PKCι and PKCζ inhibitor. CRT0066854 was able to restore polarized morphogenesis in the dysplastic H-Ras spheroids.

Pack Size	Price	Availability	Quantity
50 mg	$779	1-2 weeks
100 mg	$1,240	1-2 weeks

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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity

Description	CRT-0066854 is a PKCι and PKCζ inhibitor. CRT0066854 was able to restore polarized morphogenesis in the dysplastic H-Ras spheroids.
Targets&IC50	PKCζ:639 nM (IC50), ROCK2:620 nM (IC50)
Alias	CRT-0066854, CRT0066854, CRT 0066854

Chemical Properties

Molecular Weight	415.55
Formula	C₂₄H₂₅N₅S
Cas No.	1438881-19-6
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

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Keywords

CRT0066854 HCl