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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $95 | In Stock | |
5 mg | $356 | In Stock | |
10 mg | $533 | In Stock | |
25 mg | $863 | In Stock | |
50 mg | $1,190 | In Stock | |
100 mg | $1,580 | In Stock |
Description | ELA-14(human) acetate is a fragment of ELA that binds to APJ, activates the Gαi1 and β-arrestin-2 signaling pathways, and induces receptor internalization similarly to its parent endogenous peptide. |
In vitro | ELA-14 activates the Gαi1 and β-arrestin-2 signaling pathways with EC50s of 8.6 nM and 166 nM. ELA-14 induces receptor internalization and reduces arterial pressure, exerts positive inotropic effects on the heart[1]. |
In vivo | ELA-14 is rapidly metabolized in rat plasma (t1/2<2 min)[1]. |
Alias | ELA-14(human) acetate (1886973-05-2 free base) |
Molecular Weight | 1767.09 |
Formula | C77H123N25O19S2 |
Cas No. |
Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
Solubility Information | H2O: 100 mg/ml (56.59 mM), Sonication is recommended. ![]() | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
H2O
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