Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM). |
Targets&IC50 | mGlu4:79 nM (EC50) |
In vitro | Foliglurax is a highly selective and potent mGlu4 receptor PAM. It has a marked brain-penetrance feature, which might revolutionize the field of mGlu4 receptor drug targeting in CNS disorders [2]. |
Synonyms | PXT002331 |
Molecular Weight | 421.51 |
Formula | C23H23N3O3S |
CAS No. | 1883329-51-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5.2 mg/mL (12.34 mM), sonification/heating is recommended.
You can also refer to dose conversion for different animals. More
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Foliglurax 1883329-51-8 Neuroscience GluR PXT 002331 PXT-002331 PXT002331 inhibitor inhibit