Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2). Displays no activity at GlyT1 or 56 other common biological targets (≥ 100 μM), in a glycine uptake assay in CHO cells.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 97.00 | |
2 mg | In stock | $ 168.00 | |
5 mg | In stock | $ 217.00 | |
10 mg | In stock | $ 315.00 | |
25 mg | In stock | $ 529.00 | |
50 mg | In stock | $ 768.00 | |
100 mg | In stock | $ 1,080.00 |
Description | Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2). Displays no activity at GlyT1 or 56 other common biological targets (≥ 100 μM), in a glycine uptake assay in CHO cells. |
Targets&IC50 | GlyT2:16 nM(human) |
Molecular Weight | 448.983 |
Formula | C24H33ClN2O4 |
CAS No. | 495076-64-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 8 mg/mL
DMSO: 40 mg/mL
You can also refer to dose conversion for different animals. More
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Org 25543 hydrochloride 495076-64-7 Neuroscience GlyT Org 25543 Hydrochloride inhibitor inhibit