Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PROTAC EED degrader-1 is a PROTAC targeting EED (pKD = 9.02), is a inhibitor of polycomb repressive complex 2 (PRC2) with pIC50 of 8.17.
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Description | PROTAC EED degrader-1 is a PROTAC targeting EED (pKD = 9.02), is a inhibitor of polycomb repressive complex 2 (PRC2) with pIC50 of 8.17. |
In vitro | PROTAC EED degrader-1 binds to EED (pKD of 9.02±0.09) and inhibits PRC2 function (pIC50 of 8.17±0.24), and inhibit proliferation of an EZH2 mutant DLBCL cell line Karpas422[1]. |
Molecular Weight | 1054.2 |
Formula | C55H60FN11O8S |
CAS No. | T12553 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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PROTAC EED degrader-1 T12553 Others PROTAC EED degrader 1 PROTAC EED degrader1 inhibitor inhibit