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Adrenomedullin (AM) (22-52), human acetate
Catalog No. TP1257L
Alias Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base）
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an adrenomedullin receptor.
Adrenomedullin (AM) (22-52), human acetate
Catalog No. TP1257LAlias Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base）
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an adrenomedullin receptor.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $221 | In Stock | |
| 5 mg | $869 | In Stock | |
| 10 mg | $1,297 | In Stock | |
| 25 mg | $2,347 | In Stock |
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Purity:99.42%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an adrenomedullin receptor. |
| In vitro | Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base） competitively inhibits the binding of the Adrenomedullin dose-dependently and inhibits Adrenomedullin -induced cAMP accumulation in rat vascular smooth muscle cells. Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base） (30 nmol) selectively and reversibly decreases vasodilator responses to human calcitonin generelated peptide (hCGRP) with similar effect to that of CGRP antagonist[1]. |
| Alias | Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base） |
| Molecular Weight | 3636.09 |
| Formula | C161H256N46O50 |
Storage & Solubility Information
| Storage | store at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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