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GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $2,570 | 3-6 months | |
50 mg | $3,380 | 3-6 months | |
100 mg | $4,600 | 3-6 months |
Description | GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM). |
Targets&IC50 | GRK5:7.1 μM, GRK2:30 nM |
In vitro | GRKs-IN-1 (Compound 14as) is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine. |
Alias | GRK2-IN-1 |
Molecular Weight | 452.48 |
Formula | C24H25FN4O4 |
Cas No. | 2055990-90-2 |
Relative Density. | 1.314 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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