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CEP-28122 mesylate salt

Catalog No. T72317

CEP-28122 mesylate salt, a diaminopyrimidine derivative, is a potent, selective, and orally bioavailable ALK (anaplastic lymphoma kinase) inhibitor with an IC50 value of 1.9 nM against recombinant ALK kinase activity. It shows antitumor efficacy in ALK-positive human cancer models and has favorable pharmacodynamic and pharmacokinetic profiles.

CEP-28122 mesylate salt
Other Forms of CEP-28122 mesylate salt:
CEP-28122T26121022958-60-6
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CEP-28122 mesylate salt (1022958-60-6 free base)T10759
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CEP-28122 mesylate salt

Catalog No. T72317
CEP-28122 mesylate salt, a diaminopyrimidine derivative, is a potent, selective, and orally bioavailable ALK (anaplastic lymphoma kinase) inhibitor with an IC50 value of 1.9 nM against recombinant ALK kinase activity. It shows antitumor efficacy in ALK-positive human cancer models and has favorable pharmacodynamic and pharmacokinetic profiles.
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2 mg$985 days
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Product Introduction

Bioactivity
Description
CEP-28122 mesylate salt, a diaminopyrimidine derivative, is a potent, selective, and orally bioavailable ALK (anaplastic lymphoma kinase) inhibitor with an IC50 value of 1.9 nM against recombinant ALK kinase activity. It shows antitumor efficacy in ALK-positive human cancer models and has favorable pharmacodynamic and pharmacokinetic profiles.
Chemical Properties
Molecular Weight635.17
FormulaC29H39ClN6O6S
Storage & Solubility Information
StorageShipping with blue ice.

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