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Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $1,520 | 6-8 weeks | |
50 mg | $1,980 | 6-8 weeks | |
100 mg | $2,500 | 6-8 weeks |
Description | Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor. |
In vitro | Fosnetupitant shows a micromolar affinity for the 5-HT6 (pKi ~ 5.2) receptor and type L Ca2+ channels (pKi ~ 5.7). However, it does not bind all the other proteins investigated. |
In vivo | After i.v. injection in rats, Pronetupitant is rapidly and extensively converted to Netupitant. |
Alias | Pronetupitant |
Molecular Weight | 688.6 |
Formula | C31H35F6N4O5P |
Cas No. | 1703748-89-3 |
Relative Density. | no data available |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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